Koob · Annals of the New York Academy of Sciences 2000 · narrative review · n=?

Neurobiology of addiction. Toward the development of new therapies.

Cited 324 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review and mechanistic reasoning without new human empirical data

PubMed 10911930 · doi:10.1111/j.1749-6632.2000.tb06682.x · record verified 2026-08-31

What was done

This narrative review synthesizes neurobiological evidence and theoretical frameworks concerning the mechanisms that mediate the transition from initial drug use to compulsive drug addiction, focusing on brain circuits of positive and negative reinforcement.

What was found

The abstract reports no empirical numbers or statistical results. It outlines that acute drug reinforcement relies on the extended amygdala (including the nucleus accumbens and amygdala) and neurotransmitters including dopamine, opioid peptides, serotonin, GABA, and glutamate. Drug withdrawal engages the corticotropin-releasing factor stress system, producing reward dysregulation and an allostatic set-point shift that promotes craving and relapse vulnerability.

Why it matters

It provides a conceptual and neurochemical basis to guide rational target discovery for pharmacotherapies aimed at preventing addiction relapse.

Limits

The paper provides narrative mechanistic theory without original quantitative data, human clinical trial testing, or systematic review methodology.

Cited by