Pierre · Journal of neurochemistry 2005 · narrative review · n=?

Monocarboxylate transporters in the central nervous system: distribution, regulation and function.

Cited 731 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review of preclinical and mechanistic studies without systematic methodology

PubMed 15953344 · doi:10.1111/j.1471-4159.2005.03168.x · record verified 2026-08-30

What was done

This narrative review summarizes evidence on the regional and cellular distribution, translational regulation, and functional roles of monocarboxylate transporters (MCTs)—specifically isoforms MCT1, MCT2, and MCT4—in the mammalian and rodent central nervous system.

What was found

The abstract reports no numerical data. Qualitatively, three MCT isoforms demonstrate distinct cellular localization in rodent brain: MCT1 is expressed in microvascular endothelial cells, ependymocytes, and astrocytes; MCT4 is specific to astrocytes; and MCT2 is the predominant neuronal transporter, with immunoreactivity detected at postsynaptic sites. The review also notes that MCT expression changes across development, responds to nutritional modifications, and is regulated translationally by neurotransmitters.

Why it matters

Elucidating cell-specific MCT localization clarifies how alternative fuels like lactate, pyruvate, and ketone bodies support cerebral energetics, synaptic transmission, and metabolic homeostasis in central nervous system disorders such as ischaemia and neurodegenerative diseases.

Limits

This is a non-systematic narrative review based primarily on preclinical rodent and cellular models. The abstract presents no quantitative effect sizes, statistical metrics, search criteria, or human clinical data.

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