Surdacki · Cardiovascular & hematological agents in medicinal chemistry 2008 · narrative review · n=?

L-arginine analogs--inactive markers or active agents in atherogenesis?

Cited 33 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review synthesizing mechanistic and observational literature without systematic methodology.

PubMed 18855643 · doi:10.2174/187152508785909429 · record verified 2026-08-30

What was done

The authors reviewed literature examining the biological activities and clinical associations of the dimethylated L-arginine analogs asymmetric dimethylarginine (ADMA) and symmetric dimethylarginine (SDMA) in endothelial dysfunction, atherogenesis, and cardiovascular disease across clinical cohorts and in vitro models.

What was found

The abstract reports qualitative narrative findings without specific numerical data. ADMA levels were reported to correlate with endothelial dysfunction, atherosclerotic risk factors, and the severity of carotid, coronary, and peripheral atherosclerosis, while predicting adverse outcomes in end-stage renal disease and coronary artery disease. In vitro, proinflammatory cytokines and oxidized LDL increased endothelial ADMA release. ADMA accelerated endothelial replicative senescence via telomerase inhibition and impaired endothelial progenitor cell mobilization. SDMA was described as actively inhibiting nitric oxide synthesis by competing with endothelial L-arginine uptake.

Why it matters

This review highlights methylated arginine derivatives as active pathogenetic drivers of vascular damage and senescence rather than inert biomarkers.

Limits

As a narrative review, it lacks systematic search methodology, meta-analytic pooling, and risk-of-bias evaluation. The abstract provides no quantitative effect sizes, confidence intervals, sample sizes, or cohort details.

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