Portincasa · Current medicinal chemistry 2009 · narrative review · n=?

Medicinal treatments of cholesterol gallstones: old, current and new perspectives.

Cited 61 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review with mechanism-based reasoning and no primary data or systematic search methodology

PubMed 19355905 · doi:10.2174/092986709787909631 · record verified 2026-08-29

What was done

This narrative review summarizes medical management strategies for cholesterol gallstone disease, focusing on patient selection criteria for oral litholysis with ursodeoxycholic acid and reviewing experimental mechanisms involving intestinal cholesterol absorption inhibition (ezetimibe via NPC1L1) and nuclear receptor modulation.

What was found

The abstract reports no quantitative data or numerical outcomes. It describes that non-surgical therapy is restricted to a small subset of patients with mild symptoms and small, radiolucent, cholesterol-enriched stones inside a functioning gallbladder with a patent cystic duct. It notes that ursodeoxycholic acid acts by desaturating biliary cholesterol and that ezetimibe and nuclear receptor modulators demonstrate potential in preclinical models and preliminary human studies.

Why it matters

It outlines the narrow clinical indications where non-surgical management remains an alternative to cholecystectomy and highlights emerging molecular targets for pharmacological prevention and treatment of cholesterol gallstones.

Limits

As a narrative review, it lacks a systematic search strategy, quality appraisal of included studies, and quantitative synthesis. The abstract provides no primary human trial data, sample sizes, or precise therapeutic efficacy rates.

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