Valko · Archives of toxicology 2016 · narrative review · n=?

Redox- and non-redox-metal-induced formation of free radicals and their role in human disease.

Cited 1025 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review synthesizing biochemical and mechanistic concepts without systematic search criteria or primary empirical human data.

PubMed 26343967 · doi:10.1007/s00204-015-1579-5 · record verified 2026-08-31

What was done

This narrative review synthesizes biochemical mechanisms through which redox-active metals (iron, copper) and redox-inactive metals or metalloids (arsenic, cadmium, zinc) induce reactive oxygen species (ROS) and reactive nitrogen species (RNS). It examines the resulting oxidative damage to lipids, proteins, and DNA, as well as downstream links to chronic human pathologies.

What was found

The abstract provides no quantitative data or effect sizes. It details qualitative pathways: redox-active iron and copper undergo redox-cycling via the Fenton reaction to generate hydroxyl radicals, whereas redox-inactive arsenic and cadmium primarily exert toxicity by binding protein sulfhydryl groups and depleting glutathione. Zinc depletion impairs DNA repair mechanisms. These mechanisms cause lipid peroxidation (yielding malondialdehyde and 4-hydroxynonenal), compromise cellular antioxidant defenses (including SOD, catalase, and glutathione peroxidase), and impair signal transduction and tumor suppressor functions.

Why it matters

It provides a conceptual overview of the molecular pathways linking environmental or metabolic metal dysregulation to oxidative stress and major diseases, including cancer, cardiovascular disease, Alzheimer's disease, and Parkinson's disease.

Limits

The abstract reports no primary clinical data, quantitative risk estimates, exposure thresholds, or systematic literature search methodology. Causal links to human diseases are described at a conceptual and mechanistic level without evaluating confounding variables or clinical trial outcomes.

Cited by