Feldman · International journal of molecular sciences 2016 · narrative review · n=?

Heart Disease in Women: Unappreciated Challenges, GPER as a New Target.

Cited 21 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review synthesizing mechanistic reasoning and prior observational findings

PubMed 27213340 · doi:10.3390/ijms17050760 · record verified 2026-08-29

What was done

This narrative review describes the clinical challenges of heart disease in women, the biological basis for postmenopausal atherosclerotic risk, and evidence on the role of the G protein-coupled estrogen receptor (GPER) and its genetic variants in blood pressure and low-density lipoprotein (LDL) receptor regulation.

What was found

No quantitative data, sample sizes, or numerical effect sizes are reported in the abstract. The authors report qualitatively that GPER activation regulates blood pressure and LDL receptor metabolism, and that expression of a hypofunctional GPER variant contributes to hypertension and hypercholesterolemia, predominantly in women.

Why it matters

It highlights GPER signaling as a potential biological mechanism and therapeutic target underlying sex-specific cardiovascular risk in postmenopausal women.

Limits

As a narrative review, it lacks a systematic search strategy, quality appraisal, and meta-analytic synthesis. The abstract provides no specific numbers, effect sizes, or participant counts.

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