Sigalos · Sexual medicine reviews 2018 · Narrative review · n=?

The Safety and Efficacy of Growth Hormone Secretagogues.

Cited 45 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative literature review without systematic review methodology

PubMed 28400207 · doi:10.1016/j.sxmr.2017.02.004 · record verified 2026-08-26

What was done

The authors conducted a narrative literature review of clinical studies evaluating the safety and efficacy of growth hormone secretagogues (GHSs), including growth hormone-releasing peptides and the oral agent ibutamoren mesylate, in human subjects.

What was found

The abstract reports no quantitative figures or statistical values. GHSs stimulate pulsatile growth hormone secretion that remains subject to normal negative feedback mechanisms. Qualitatively, reviewed evidence suggests GHSs can improve growth velocity in children, stimulate appetite, enhance fat-free and lean mass in obesity and wasting conditions, reduce bone turnover, and improve sleep. GHSs were generally well tolerated, with potential adverse increases in blood glucose driven by reduced insulin sensitivity.

Why it matters

Exogenous growth hormone carries risks related to supra-therapeutic levels and disrupted feedback loops. GHSs represent an alternative therapeutic approach that may preserve endogenous physiological regulation, though clinical adoption requires clearer risk-benefit validation.

Limits

The abstract presents no quantitative data, effect sizes, or meta-analytic pooling. The underlying literature contains few long-term, rigorously controlled clinical trials, and critical long-term safety outcomes—such as cancer incidence, cardiovascular effects, and mortality—remain unmeasured.

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