Mayer · The Annals of pharmacotherapy 2020 · systematic review · n=4 studies

Bremelanotide: New Drug Approved for Treating Hypoactive Sexual Desire Disorder.

Cited 45 times in the scientific literature.

Level 1 - systematic review of randomized trials

Systematic review of phase 2 and phase 3 clinical trials

PubMed 31893927 · doi:10.1177/1060028019899152 · record verified 2026-08-29

What was done

A systematic review of literature from Medline, SCOPUS, and EMBASE (January 1, 1996, to December 15, 2019) evaluating bremelanotide for hypoactive sexual desire disorder (HSDD). The authors extracted data from 2 phase 3 trial reports and 2 phase 2 trial reports, along with supplementary analyses.

What was found

Bremelanotide demonstrated statistically significant improvements in sexual desire and reductions in distress related to lack of desire, though the authors note the clinical benefit may be modest. The most common adverse effects were nausea (39.9%), facial flushing (20.4%), and headache (11%). Absolute numerical change scores and confidence intervals for efficacy endpoints were not reported in the abstract.

Why it matters

As the second FDA-approved therapy for HSDD, as-needed subcutaneous bremelanotide offers an option with limited drug-drug interactions and no significant ethanol interaction, though clinicians must weigh modest clinical benefits against frequent nausea.

Limits

The abstract synthesizes only 4 trial reports and omits exact participant counts, baseline characteristics, and numerical efficacy outcome data (e.g., scale scores or effect sizes). Long-term adherence given high nausea rates and comparative effectiveness against other therapies were not detailed in the abstract.

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