Andres-Hernando · JCI insight 2021 · preclinical animal and mechanistic study · n=?

Vasopressin mediates fructose-induced metabolic syndrome by activating the V1b receptor.

Cited 55 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Preclinical animal model and mechanistic laboratory study

PubMed 33320834 · doi:10.1172/jci.insight.140848 · record verified 2026-08-27

What was done

The authors investigated whether vasopressin mediates fructose-induced metabolic syndrome. Mice were administered oral fructose, glucose, or high-fructose corn syrup to assess copeptin (vasopressin surrogate) responses and fructokinase involvement. The effects of suppressing vasopressin via increased hydration were tested, and knockout mouse models (V1bR-KO and V1a-KO) were evaluated alongside measurements of hepatic V1bR and fructokinase expression.

What was found

The abstract reports no numerical values. Qualitatively, oral sugar intake elevated copeptin levels in a fructokinase-dependent manner. Vasopressin suppression via hydration both prevented and ameliorated metabolic syndrome. V1bR-KO mice were completely protected from fructose-induced metabolic syndrome, whereas V1a-KO mice exhibited worsened metabolic syndrome. Fructose ingestion induced de novo hepatic V1bR expression, which in turn amplified fructokinase expression.

Why it matters

This work outlines a mechanistic link between water conservation pathways and fat accumulation, identifying the vasopressin V1b receptor as a mediator of fructose-induced metabolic dysfunction. It offers a mechanistic rationale for testing increased water intake in human metabolic disease.

Limits

All findings are derived from preclinical mouse models with no human clinical data. The abstract provides no specific sample sizes, sugar dosages, treatment durations, or quantitative effect sizes.

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