Hardeland · Antioxidants & redox signaling 2022 · narrative review · n=?

Redox Biology of Melatonin: Discriminating Between Circadian and Noncircadian Functions.

Cited 64 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review of biological mechanisms without original human data or systematic review methodology.

PubMed 35018802 · doi:10.1089/ars.2021.0275 · record verified 2026-08-31

What was done

This narrative review synthesized literature differentiating the circadian chronobiotic roles of melatonin from its noncircadian protective actions. The authors evaluated mechanisms involving extrapineal synthesis, mitochondrial formation, sirtuin upregulation, microRNA regulation, and the modulation of inflammation and oxidative stress.

What was found

The abstract reports no numerical data or statistical effect sizes. It describes qualitative mechanistic distinctions showing that noncircadian melatonin functions provide mitochondrial protection, antioxidant defense, and anti-inflammatory effects (including macrophage/microglia polarization and avoidance of cytokine storms) with signaling pathways and dose requirements distinct from circadian regulation.

Why it matters

Distinguishing chronobiotic actions from direct cytoprotective mechanisms provides a theoretical basis for evaluating high-dose melatonin in acute inflammatory and mitochondrial-related diseases, including severe infections.

Limits

This is a narrative review without systematic search criteria or original empirical data. The abstract provides no quantitative metrics, human clinical trial data, or specific dosage thresholds.

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