García-Villalba · Molecular nutrition & food research 2022 · narrative review · n=?

Urolithins: a Comprehensive Update on their Metabolism, Bioactivity, and Associated Gut Microbiota.

Cited 289 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative review of preclinical literature and preliminary human studies

PubMed 35118817 · doi:10.1002/mnfr.202101019 · record verified 2026-08-26

What was done

This review synthesized literature from the preceding five years regarding urolithins—gut microbiota-derived metabolites of ellagitannins and ellagic acid found in foods like pomegranates, walnuts, and strawberries. It examined the chemical diversity of urolithins, their tissue and fluid distribution in humans, the microbial ecology defining specific metabotypes (UM-A, UM-B, UM-0), and the bioactivity and safety profile of urolithin A across preclinical models and initial human trials.

What was found

Thirteen urolithins and their conjugated derivatives (glucuronides, sulfates) have been detected across multiple human tissues and biofluids, including urine, blood, feces, breastmilk, prostate, colon, and breast tissue. The abstract reports no numerical effect sizes or quantitative outcome statistics.

Why it matters

It organizes the current understanding of how dietary polyphenols are converted into active metabolites and highlights gut microbiome-dependent metabotypes that may explain individual variations in health responses.

Limits

The paper is a non-systematic narrative review without standardized quality appraisal or quantitative synthesis. As noted in the abstract, many published in vitro studies used non-physiological concentrations or non-conjugated molecular forms, questioning reported mechanisms, and human intervention evidence remains in early stages.

Cited by