Kreider · Nutrients 2022 · narrative critical review · n=?

Bioavailability, Efficacy, Safety, and Regulatory Status of Creatine and Related Compounds: A Critical Review.

Cited 94 times in the scientific literature.

Level 5 - mechanism / opinion, no new human data

Narrative critical review without systematic search or meta-analytic methodology.

PubMed 35268011 · doi:10.3390/nu14051035 · record verified 2026-08-26

What was done

The authors conducted a critical review summarizing the physicochemical properties, bioavailability, efficacy, safety, and regulatory status of creatine monohydrate compared to alternative marketed novel creatine forms. They categorized marketed forms by evidence strength regarding bioavailability and safety, and outlined evidentiary requirements needed to substantiate supplement claims.

What was found

The abstract reports no numerical values, statistics, or effect sizes. The authors concluded that creatine monohydrate remains the only creatine form supported by substantial evidence for bioavailability, safety, and efficacy, and that it is the primary form approved by regulatory bodies and recommended by professional organizations. Marketed alternative forms were reported to be generally less bioavailable, less effective in comparative trials, more expensive, or insufficiently studied.

Why it matters

This paper clarifies that novel and marketed alternative forms of creatine do not have superior evidence over standard creatine monohydrate for efficacy or safety.

Limits

The abstract describes a narrative critical review rather than a systematic review or meta-analysis. No quantitative metrics, search strategies, or study sample sizes are reported in the abstract.

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